Catalyst-free synthesis of fused Triazolo-Diazepino[5,6-b]Quinoline derivatives via a sequential Ugi-4CR-nucleophilic substitution-intramolecular click reaction
A convenient, post-transformational reaction has been developed for the construction of highly diversified quinoline-fused triazolo-diazepinones featuring four diversification points by employing a catalyst-free Ugi four-component-nucleophilic substitution-intramolecular click cycloaddition sequen...
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| Main Authors: | , |
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| Format: | Article (Journal) |
| Language: | English |
| Published: |
29.01.2018
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| In: |
Synlett
Year: 2018, Volume: 29, Issue: 08, Pages: 1095-1101 |
| ISSN: | 1437-2096 |
| DOI: | 10.1055/s-0036-1591531 |
| Online Access: | Verlag, Volltext: https://doi.org/10.1055/s-0036-1591531 Verlag: http://www.thieme-connect.de/DOI/DOI?10.1055/s-0036-1591531 
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| Author Notes: | Saeed Balalaie, Aref Vaezghaemi, Nahid Zarezadeh, Frank Rominger, Hamid Reza Bijanzadeh |
| Summary: | A convenient, post-transformational reaction has been developed for the construction of highly diversified quinoline-fused triazolo-diazepinones featuring four diversification points by employing a catalyst-free Ugi four-component-nucleophilic substitution-intramolecular click cycloaddition sequence. This approach provides a wide scope of products with good yields and high bond-forming efficiency. |
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| Item Description: | Gesehen am 03.03.2020 Der Buchstabe "b" ist im Titel kursiv geschrieben |
| Physical Description: | Online Resource |
| ISSN: | 1437-2096 |
| DOI: | 10.1055/s-0036-1591531 |