Concentration effect relationship of CYP3A inhibition by ritonavir in humans

To investigate the dose and concentration dependency of CYP3A inhibition by ritonavir using the established limited sampling strategy with midazolam for CYP3A activity.

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Bibliographic Details
Main Authors: Eichbaum, Christine (Author) , Cortese, Marianna (Author) , Blank, Antje (Author) , Burhenne, Jürgen (Author) , Mikus, Gerd (Author)
Format: Article (Journal)
Language:English
Published: 9 June 2013
In: European journal of clinical pharmacology
Year: 2013, Volume: 69, Issue: 10, Pages: 1795-1800
ISSN:1432-1041
DOI:10.1007/s00228-013-1530-8
Online Access:Verlag, lizenzpflichtig, Volltext: https://doi.org/10.1007/s00228-013-1530-8
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Author Notes:Christine Eichbaum, Marianna Cortese, Antje Blank, Jürgen Burhenne, Gerd Mikus
Description
Summary:To investigate the dose and concentration dependency of CYP3A inhibition by ritonavir using the established limited sampling strategy with midazolam for CYP3A activity.
Item Description:Gesehen am 08.01.2021
Physical Description:Online Resource
ISSN:1432-1041
DOI:10.1007/s00228-013-1530-8