Comparing the efficacy and selectivity of Ck2 inhibitors: a phosphoproteomics approach

CK2 (an acronym derived from the misnomer “casein kinase 2”) denotes a ubiquitous, highly pleiotropic protein kinase which has been implicated in global human pathologies, with special reference to cancer. A large spectrum of fairly selective, cell permeable CK2 inhibitors are available, one of whic...

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Main Authors: Borgo, Christian (Author) , Cesaro, Luca (Author) , Hirota, Tsuyoshi (Author) , Kuwata, Keiko (Author) , D’Amore, Claudio (Author) , Ruppert, Thomas (Author) , Blatnik, Renata (Author) , Salvi, Mauro (Author) , Pinna, Lorenzo A. (Author)
Format: Article (Journal)
Language:English
Published: 27 January 2021
In: European journal of medicinal chemistry
Year: 2021, Volume: 214, Pages: 1-11
ISSN:1768-3254
DOI:10.1016/j.ejmech.2021.113217
Online Access:Verlag, lizenzpflichtig, Volltext: https://doi.org/10.1016/j.ejmech.2021.113217
Verlag, lizenzpflichtig, Volltext: https://www.sciencedirect.com/science/article/pii/S0223523421000660
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Author Notes:Christian Borgo, Luca Cesaro, Tsuyoshi Hirota, Keiko Kuwata, Claudio D’Amore, Thomas Ruppert, Renata Blatnik, Mauro Salvi, Lorenzo A. Pinna
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