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A mild method for regioselective labeling of aromatics with radioactive iodine

A novel technique to label ortho-, meta-, and para-trimethylsilyl-substituted aryl substituents with radioactive iodide is described. The method takes advantage of the ipso-directing and activating properties of trimethylsilyl substituents on the arenes. The method was demonstrated on a griseofulvin...

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Hauptverfasser: Rønnest, Mads H. (VerfasserIn) , Nissen, Felix (VerfasserIn) , Pedersen, Palle J. (VerfasserIn) , Larsen, Thomas O. (VerfasserIn) , Mier, Walter (VerfasserIn) , Clausen, Mads H. (VerfasserIn)
Dokumenttyp: Article (Journal) Editorial
Sprache:Englisch
Veröffentlicht: May 14, 2013
In: European journal of organic chemistry
Year: 2013, Heft: 19, Pages: 3970-3973
ISSN:1099-0690
DOI:10.1002/ejoc.201300419
Online-Zugang:Verlag, lizenzpflichtig, Volltext: https://doi.org/10.1002/ejoc.201300419
Verlag, lizenzpflichtig, Volltext: https://onlinelibrary.wiley.com/doi/abs/10.1002/ejoc.201300419
Volltext
Verfasserangaben:Mads H. Rønnest, Felix Nissen, Palle J. Pedersen, Thomas O. Larsen, Walter Mier, and Mads H. Clausen

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