First fluorescent acetylspermidine deacetylation assay for HDAC10 identifies selective inhibitors with cellular target engagement
HDAC, histone deacetylases, HDAC10, medicinal chemistry, polyamines
Gespeichert in:
| Hauptverfasser: | , , , , , , , , , , , , , , , , , |
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| Dokumenttyp: | Article (Journal) |
| Sprache: | Englisch |
| Veröffentlicht: |
July 19, 2022
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| In: |
ChemBioChem
Year: 2022, Jahrgang: 23, Heft: 14, Pages: 1-28 |
| ISSN: | 1439-7633 |
| DOI: | 10.1002/cbic.202200180 |
| Online-Zugang: | Resolving-System, kostenfrei: https://doi.org/10.1002/cbic.202200180 Resolving-System, kostenfrei: https://doi.org/10.25673/101612 
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| Verfasserangaben: | Daniel Herp, Johannes Ridinger, Dina Robaa, Stephen A. Shinsky, Karin Schmidtkunz, Talha Z. Yesiloglu, Theresa Bayer, Raphael R. Steimbach, Corey J. Herbst-Gervasoni, Annika Merz, Christophe Romier, Peter Sehr, Nikolas Gunkel, Aubry K. Miller, David W. Christianson, Ina Oehme, Wolfgang Sippl, and Manfred Jung |
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