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Interaction potential of etravirine with drug transporters assessed in vitro

Etravirine is a novel nonnucleoside reverse transcriptase inhibitor (NNRTI) for the treatment of HIV-1 infections. ABC transporters potentially mediate clinically relevant drug-drug interactions. We assessed substrate characteristics and the inhibitory and inductive potential of etravirine on ABC tr...

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Hauptverfasser: Zembruski, Nadine Cécile Luise (VerfasserIn) , Haefeli, Walter E. (VerfasserIn) , Weiß, Johanna (VerfasserIn)
Dokumenttyp: Article (Journal)
Sprache:Englisch
Veröffentlicht: February 24, 2011
In: Antimicrobial agents and chemotherapy
Year: 2011, Jahrgang: 55, Heft: 3, Pages: 1282-1284
ISSN:1098-6596
DOI:10.1128/AAC.01527-10
Online-Zugang:Verlag, lizenzpflichtig, Volltext: https://doi.org/10.1128/AAC.01527-10
Verlag, lizenzpflichtig, Volltext: https://journals.asm.org/doi/10.1128/AAC.01527-10
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Verfasserangaben:Nadine Cécile Luise Zembruski, Walter Emil Haefeli, and Johanna Weiss

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