Design, synthesis and biological evaluation of simplified analogues of the RNA polymerase inhibitor etnangien
Novel simplified analogues of the potent RNA polymerase inhibitor etnangien were obtained by total synthesis and evaluated for antibacterial activity against Gram-positive bacteria and one Gram-negative bacterium.
Gespeichert in:
| Hauptverfasser: | , , |
|---|---|
| Dokumenttyp: | Article (Journal) |
| Sprache: | Englisch |
| Veröffentlicht: |
2010
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| In: |
Bioorganic & medicinal chemistry letters
Year: 2010, Jahrgang: 20, Heft: 3, Pages: 939-941 |
| ISSN: | 1464-3405 |
| DOI: | 10.1016/j.bmcl.2009.12.066 |
| Online-Zugang: | Verlag, lizenzpflichtig, Volltext: https://doi.org/10.1016/j.bmcl.2009.12.066 Verlag, lizenzpflichtig, Volltext: https://www.sciencedirect.com/science/article/pii/S0960894X09017892 |
| Verfasserangaben: | Dirk Menche, Pengfei Li, Herbert Irschik |
MARC
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