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Lack of CYP3A4 protein induction despite mRNA induction in primary hepatocytes exposed to rifabutin as a possible explanation for its low interaction risk in vivo von Nilles, Julie (VerfasserIn) , Theile, Dirk (VerfasserIn) , Weiß, Johanna (VerfasserIn) , Haefeli, Walter E. (VerfasserIn) , Ruez, Stephanie (VerfasserIn) ,
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The differences in drug disposition gene induction by rifampicin and rifabutin are unlikely due to different effects on important pregnane X receptor (NR1I2) splice variants von Nilles, Julie (VerfasserIn) , Weiß, Johanna (VerfasserIn) , Masin, Martin (VerfasserIn) , Tuffs, Christopher (VerfasserIn) , Strowitzki, Moritz (VerfasserIn) , Haefeli, Walter E. (VerfasserIn) , Ruez, Stephanie (VerfasserIn) , Theile, Dirk (VerfasserIn) ,
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Ähnliche Schlagworte
Rifabutin
Rifampicin
ATP Binding Cassette Transporter, Subfamily B
ATP Binding Cassette Transporter, Subfamily B, Member 1
CYP3A4
Cells, Cultured
Cytochrome P-450 CYP3A
Cytochrome P-450 CYP3A Inducers
Drug Interactions
Enzyme Induction
Expression
Hepatocytes
Humans
Induction
Male
P-gp
Pregnane X receptor
Primary human hepatocyte
Primary human hepatocytes
RNA, Messenger
Rifampin
Splice variant
Tandem Mass Spectrometry