First fluorescent acetylspermidine deacetylation assay for HDAC10 identifies selective inhibitors with cellular target engagement

HDAC, histone deacetylases, HDAC10, medicinal chemistry, polyamines

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Bibliographic Details
Main Authors:	Herp, Daniel (Author) , Ridinger, Johannes (Author) , Robaa, Dina (Author) , Shinsky, Stephen A. (Author) , Schmidtkunz, Karin (Author) , Yesiloglu, Talha Z. (Author) , Bayer, Theresa Yasmin Charlotte (Author) , Steimbach, Raphael R. (Author) , Herbst-Gervasoni, Corey J. (Author) , Merz, Annika (Author) , Romier, Christophe (Author) , Sehr, Peter (Author) , Gunkel, Nikolas (Author) , Miller, Aubry K. (Author) , Christianson, David W. (Author) , Oehme, Ina (Author) , Sippl, Wolfgang (Author) , Jung, Manfred (Author)
Format:	Article (Journal)
Language:	English
Published:	July 19, 2022
In:	ChemBioChem Year: 2022, Volume: 23, Issue: 14, Pages: 1-28
ISSN:	1439-7633
DOI:	10.1002/cbic.202200180
Online Access:	Resolving-System, kostenfrei: https://doi.org/10.1002/cbic.202200180 Resolving-System, kostenfrei: https://doi.org/10.25673/101612
Author Notes:	Daniel Herp, Johannes Ridinger, Dina Robaa, Stephen A. Shinsky, Karin Schmidtkunz, Talha Z. Yesiloglu, Theresa Bayer, Raphael R. Steimbach, Corey J. Herbst-Gervasoni, Annika Merz, Christophe Romier, Peter Sehr, Nikolas Gunkel, Aubry K. Miller, David W. Christianson, Ina Oehme, Wolfgang Sippl, and Manfred Jung

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Summary:	HDAC, histone deacetylases, HDAC10, medicinal chemistry, polyamines
Item Description:	Published online: 24 May 2022
Physical Description:	Online Resource
ISSN:	1439-7633
DOI:	10.1002/cbic.202200180